Lipids and Lipid Derivatives
TARGETMOL CHEMICALS INC Nomegestrol acetate 25MG
Also available in 1 mL, 2 mg, 5 mg, 10 mg, 50 mg, 100 mg, 200 mg and bulk. Please contact Fisher for quotes.Nomegestrol acetate is a widely used progestin-like drug,which is characterized as a full agonist at the progesterone receptor Purity 99.93%
TARGETMOL CHEMICALS INC Alarelin Acetate 25MG
Also available in 1 mL, 5 mg, 10 mg, 50 mg, 100 mg, 500 mg and bulk. Please contact Fisher for quotes. Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
Medchemexpress LLC Incensole Acetate | 34701-53-6 | 1 MG
Incensole Acetate, a main constituent of Boswellia carterii resin, demonstrates neuroprotective effects against neuronal damage from traumatic and ischemic head injury. It has been shown to reduce Aβ25-35-triggered apoptosis in hOBNSCs and, in in vitro studies, significantly ameliorates Aβ25-35-induced cell death.
- Demonstrates neuroprotective effects against neuronal damage
- Reduces Aβ25-35-triggered apoptosis in hOBNSCs
- Ameliorates Aβ25-35-induced cell death in in vitro studies
- High purity of 99.08%
- Soluble in DMSO
Medchemexpress LLC MK2-IN-5 acetate (Hsp25 kinase inhibitor acetate) | 99.64% | 1396.68 | 10 MG
MK2-IN-5 acetate (Hsp25 kinase inhibitor acetate) is a Mk2 pseudosubstrate with a Ki of 8 μM. It targets the protein interaction domain in the MAPK pathway and inhibits HSP25 and HSP27 phosphorylation. In vitro, MK2-IN-5 acetate (5-10 μM, 2 hours) inhibits TGF-β1 induced connective tissue growth factor (CTGF) and collagen type I in primary human keloid fibroblasts. In vivo, a single intraperitoneal injection of 2 mg/kg of MK2-IN-5 acetate decreased HSP25 phosphorylation in a ventilator-associated lung injury model.
Medchemexpress LLC L57 acetate | 99.0% | 2483.87 (free base) | 10 MG
L57 acetate is a Low-density lipoprotein receptor-related protein 1 (LRP1)-binding peptide. It demonstrates a high affinity for LRP1 with a Ki of 45 nM. This peptide also exhibits blood-brain barrier (BBB) permeability and plasma stability, making it a potential carrier for central nervous system (CNS) drug delivery.
- High affinity to LRP1 (Ki of 45 nM)
- Exhibits blood-brain barrier (BBB) permeability
- Demonstrates plasma stability
- Potential as a carrier for CNS drug delivery
Medchemexpress LLC TAT-QFNP12 acetate | 3006.47 (free base) | 1 MG
TAT-QFNP12 acetate is a peptide that plays a crucial role in cellular signaling pathways. It functions by blocking the NDRG2-PPM1A binding, which in turn reduces Smad2/3 phosphorylation. This peptide is also known to decrease astrocytic MMP-9 production and mitigate blood-brain barrier (BBB) disruption following subarachnoid hemorrhage (SAH).
- Blocks NDRG2-PPM1A binding
- Reduces Smad2/3 phosphorylation
- Decreases astrocytic MMP-9 production
- Mitigates blood-brain barrier (BBB) disruption after subarachnoid hemorrhage (SAH)
Medchemexpress LLC Protirelin Acetate | 120876-23-5 | 99.9% | 452.46 | 100 MG
Protirelin Acetate is a highly conserved neuropeptide that exerts hormonal control of thyroid-stimulating hormone (TSH) levels and has neuromodulatory functions. This product is for research use only.
- Exerts hormonal control of thyroid-stimulating hormone (TSH) levels
- Has neuromodulatory functions
- Targeted to the thyroid hormone receptor
- Involved in the vitamin D related/nuclear receptor pathway
- Appears as a white to off-white solid
- Sequence: {pGlu}-His-Pro-NH2
- Sequence shortening: {pGlu}-HP-NH2
Medchemexpress LLC Protirelin acetate | 120876-23-5 | CB8947811 | 99.9% | 452.46 | 50 MG
Protirelin acetate is a highly conserved neuropeptide that exerts hormonal control of thyroid-stimulating hormone (TSH) levels and also has neuromodulatory functions.
- Exerts hormonal control of thyroid-stimulating hormone (TSH) levels
- Functions as a neuromodulator
- Targets the thyroid hormone receptor
- Stable as powder for 2 years at -80°C or 1 year at -20°C
- Stable in solvent for 6 months at -80°C or 1 month at -20°C
Medchemexpress LLC 1-O-n-Octyl-B-D-gluc 1mg | 129522-81-2 | 309.47 g·mol^-1 | C14H11D17O6 | 1 MG
Deuterated n-octyl β-D-glucopyranoside (d17) is a deuterium-labeled non-ionic detergent used to solubilize membrane proteins and as an analytical standard in quantitative methods. It is supplied in small, research-scale quantities for biochemical and analytical workflows.
- Deuterium-labeled non-ionic detergent for membrane protein solubilization.
- Serves as a tracer and internal standard for quantitative NMR, GC-MS, and LC-MS.
- Supplied in small, research-grade quantities suitable for analytical use.
- Deuteration provides a mass shift for clear distinction from unlabeled analogs in mass spectrometry.
- Batch-specific certificate of analysis available for purity and isotopic enrichment verification.
Medchemexpress LLC Bradykinin acetate | 6846-03-3 | 99.6% | 1060.21 (free base) | 100 MG
Bradykinin acetate | 6846-03-3 | 99.6% | 1060.21 (free base) | 100 MG
Medchemexpress LLC Larazotide (acetate) | 881851-50-9 | MFCD31630844 | 99.7% | 785.89 g/mol | C34H59N9O12 | 100 MG
Larazotide acetate is an eight-amino-acid peptide zonulin antagonist supplied as a research reagent. It is used in studies of celiac disease and intestinal barrier dysfunction and has reported antiviral activity against varicella-zoster virus. For research use only; not for human therapeutic use.
- Eight-amino-acid peptide sequence: Gly-Gly-Val-Leu-Val-Gln-Pro-Gly.
- Orally active zonulin antagonist that modulates tight junctions.
- Reported in vitro antiviral activity versus varicella-zoster virus.
- Supplied as a powder; recommended sealed, cold storage to preserve stability.
- Well characterized molecular weight and formula for research applications.
Medchemexpress LLC PNC-27 acetate | 99.98% | 4031.73 (free base) | 100 MG
PNC-27 acetate is a chimeric p53-penetratin peptide that binds to HDM-2 in a p53 peptide-like structure.
- Induces selective membrane-pore formation, leading to cancer cell lysis.
- Utilized in acute myeloid leukemia research.
Medchemexpress LLC Iso-VQA-ACC acetate | 99.48% | 625.63 (free base) | 1 MG
iso-VQA-ACC acetate is a substrate for constitutive proteasome, characterized by its molecular formula C29H35N7O9.xC2H4O2 and a molecular weight of 625.63 (free base). This compound has a purity of 99.48% and is commonly identified by its sequence, iso-Val-Gln-Ala-{ACC}. It is primarily used in research involving proteasome and metabolic enzyme/protease pathways.
- Targets proteasome activity for metabolic studies.
- High purity suitable for sensitive research applications.
- Soluble in DMSO at 100 mg/mL, requiring ultrasonic treatment for dissolution.
Medchemexpress LLC KRpTIRR acetate | 98.2% | 908.99 | 1 MG
KRpTIRR acetate is a phosphothreonine-containing peptide that serves as a substrate for phosphatases.
- Appearance: Solid, white to off-white
- Sequence: Lys-Arg-{Thr
}-Ile-Arg-Arg (KR-{Thr }-IRR) - Solubility in water: Greater than or equal to 100 mg/mL
- Functions as a peptide, enzyme substrate, and phosphatase inhibitor